5
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6134 | IEM 1754 2HBr | IEM 1754 dihydrobromide | GluR |
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM. | |||
T70922 | SKF32802 | ||
SKF32802 is a novel potent, selective hERG potassium channel (Kv11.1) activator that induces a leftward shift in the voltage dependence of activation. | |||
T70691 | ITP-2 | ||
ITP-2 is a selective activator of hERG channels. ITP-2 causes large depolarizing shifts in the midpoint of voltage-dependent inactivation and hyperpolarizing shifts in the voltage-dependence of activation. | |||
TP1531 | Guangxitoxin 1E | ||
Guangxitoxin 1E acts as a gating modifier since it shifts the voltage-dependence of Kv2.1 K+ currents towards depolarized potentials. | |||
T80638 | Glycinexylidide | GX | MEK |
Glycinexylidide (GX), the active metabolite of the local anesthetic Lidocaine, exhibits properties significant in inhibiting sodium channels with complex voltage dependence and mitigates the proliferation and spread of g... |